Bromosporine ≥98% (by HPLC)

Synonyms: Ethyl (3-methyl-6-(4-methyl-3-(methylsulfonamido)phenyl)-[1,2,4]triazolo[4,3-b]pyridazin-8-yl)carbamateEthyl (3-methyl-6-(4-methyl-3-(methylsulphonamido)phenyl)-[1,2,4]triazolo[4,3-b]pyridazin-8-yl)carbamate

2652-5 2652-1
76021-368EA 87.57 USD
76021-368 76021-370
Bromosporine ≥98% (by HPLC)
Bromosporine

Bromosporine is a broad spectrum bromodomain inhibitor (IC₅₀s = 0.41 µM, 0.29 µM, 0.122 µM and 0.017 µM for BRD2, BRD4, BRD9 and CECR2, respectively). At 1 µM, Bromosporine accelerates FRAP recovery of BRD4 and CREBBP, while displaying no activities against TIF1α, BAZ2A, and SMARCA2 even at 10 µM.

Formula: C₁₇H₂₀N₆O₄S
MW: 404.44 g/mol
Storage Temperature: Freezer
MDL Number: MFCD26142669
CAS Number: 1619994-69-2
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