I-BET762 ≥98% (by HPLC)

Synonyms: 2-((4S)-6-(4-Chlorophenyl)-8-methoxy-1-methyl-4H-benzo[f][1,2,4]triazolo[4,3-a][1,4]diazepin-4-yl)-N-ethylacetamideGSK525762(4S)-6-(4-Chlorophenyl)-N-ethyl-8-methoxy-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepine-4-acetamide

2628-5 2628-1
76021-282EA 99.24 USD
76021-282 76021-284
I-BET762 ≥98% (by HPLC)
I-BET762

I-BET762 (GSK525762) is a highly potent, selective and cell-permeable inhibitor of the bromodomain and extra terminal (BET) family protein BRD4 (IC₅₀ of ~35 nM). It inhibits myeloma cell proliferation and suppresses the production of proinflammatory proteins by macrophages and blocks acute inflammation.


  • Appearance: Off-white solid

Formula: C₂₂H₂₂ClN₅O₂
MW: 423.9 g/mol
Storage Temperature: Freezer
MDL Number: MFCD22417091
CAS Number: 1260907-17-2
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