Gabexate mesylate ≥98% (by HPLC)

Supplier: Enzo Life Sciences

Synonyms: 4-[[6-[(Aminoiminomethyl)amino]-1-oxohexyl]oxy]benzoic acid ethyl ester MesylateGabexate MethanesulphonateEthyl 4-((6-guanidinohexanoyl)oxy)benzoate methanesulphonateGabexate MethanesulfonateEthyl 4-((6-guanidinohexanoyl)oxy)benzoate methanesulfonate

BML-PI144-0050 BML-PI144-0010
89161-682EA 108.66 USD
89161-682 89161-684
Gabexate mesylate ≥98% (by HPLC)
Gabexate mesylate

A competitive, reversible inhibitor of serine proteases tryptase (Ki=3.4nM), thrombin (Ki=500nM), uPA (Ki=1.3µM), plasmin (Ki=1.5µM), trypsin (Ki=2µM), factor Xa (Ki=2µM). At higher concentrations it inhibits kallikrein-1 (Ki=2.6mM), C1 esterase (IC50=520µM), as well as phospholipase A2 (IC50=500µM), rat iNOS (Ki=5mM) and cNOS (Ki=150µM), and swine kidney copper amine oxidase (Ki=27µM), but not chymotrypsin. Has been used in tissue culture and in vivo. In clinical use for pancreatitis.


  • Protease inhibitor


White solid.


Soluble in water (25 mg/ml).

Formula: C₁₆H₂₃N₃O₄·CH₃SO₃H
MW: 417.5 g/mol
Storage Temperature: Freezer
MDL Number: MFCD00210299
CAS Number: 56974-61-9

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